Hormones are chemical messengers that initiate fundamental changes in the body. One such hormone, testosterone, is found in humans, as well as in other animals. Later on, in this article, we will go over the most Effective Testosterone Blockers
Testosterone is the primary hormone responsible for many of the physical characteristics peculiar to individuals with testes. It belongs to a class of male hormones called androgens, also called steroids or anabolic steroids.
It fuels the development of male sex organs before birth, even the development and maintenance of masculine secondary sex characteristics, including a deep voice, broad shoulders, growth of facial and body hair, and muscle and fat distribution.
The testicles principally produce testosterone in men while the ovaries do so in women but much smaller amounts. Testosterone levels in women are a tenth to a twentieth of men’s levels.
The adrenal glands also produce small quantities of testosterone in both sexes. Testosterone levels are highest by age 20 to 30 and slowly begin to decrease after age 30 to 35.
Testosterone controls the appearance and sexual development and is essential for the production of sperm in adult life.
It builds bone and muscle mass, increases body and pubic hair growth, height, enlargement of the penis, testes and prostate gland, and changes sexual and aggressive conduct.
To produce these changes; testosterone is converted into another androgen known as dihydrotestosterone (DHT). Testosterone is synthesized in the body from cholesterol.
The brain’s hypothalamus and pituitary gland regulate testosterone production. The brain, through chemicals and hormones in the bloodstream, signals the pituitary gland, which then relays signals to the testes to produce testosterone or decrease its production.
Not all transfeminine individuals wish to undertake a medical or surgical gender change, though many do. An objective of transgender medical intervention is to align physical characteristics with gender identity.
For some transgender individuals, having a body that more closely matches their gender identity can decrease discomfort. The first step usually is to begin cross-sex hormone therapy.
This is where testosterone blockers come in.
Testosterone blockers block the action of testosterone in your body and prevent the production of testosterone. For transgender women, hormone therapy involves not only the use of estrogen or estradiol but also the use of a testosterone blocker as well because testosterone acts much more strongly than estrogen does.
There are several physical differences between men and women that are sex-linked and are caused by differences in testosterone and estrogen.
Some developmental changes take place differently and are contingent on whether testosterone or estrogen is dominant in the body. Testosterone is more efficient at masculinizing someone than estrogen is at feminizing a person.
This makes transitioning more difficult for transgender women. They cannot rely on estrogen alone for the development of more feminine characteristics.
They must adjunctively lower their average testosterone concentrations. Testosterone Blockers have proven successful in achieving this goal.
Two testosterone blockers commonly used for transgender women are spironolactone and cyproterone acetate. Evidence indicates that spironolactone is a very safe way to lower testosterone, but is the prescription process is difficult for most.
Testosterone blockers are anti-androgens. An anti-androgen is a compound that has the biological effect of blocking or repressing the action of male sex hormones within the human body.
Testosterone blockers prevent the effects of testosterone and DHT in the body. They act by blocking them from binding to and activating the androgen receptor.
They also work to suppress the production of androgens. Anti-testosterone treatments such as spironolactone and cyproterone are successful therapies, given in addition to estrogen, to reduce testosterone concentrations to the typical female levels.
The addition of testosterone blockers to estrogen therapy is often necessary to lower testosterone values to the feminine scale.
Good Testosterone Blockers also work by reducing the secretion of luteinizing hormone and follicle-stimulating hormone; this leads to reduced stimulation of testicular testosterone production.
Testosterone blockers could be started before estrogen, or taken together. They will block the effects of testosterone and also reduce its levels in the bloodstream.
With the changes in testosterone levels come noticeable changes such as:
Slowing of baldness
Softer skin and hair
Breast development and tenderness
Change in body fat distribution
A decrease in testicular size
Lowered sexual desires and function
Decreased facial hair growth
“Testosterone blockers” can gradually bring about such changes in 6 to 12 months, but its effects may vary from person to person. Testosterone blockers, together with estrogen, can help to both suppress masculine traits and promote feminine ones.
Most testosterone blockers are very safe, but they may have side effects. The prescription testosterone blocker most often used, spironolactone, for example, can cause you to urinate overly and feel lightheaded, particularly when you first start taking it.
It is essential to drink lots of fluids with this treatment. Spironolactone can prove dangerous for people with kidney and blood pressure problems.
It is essential to consult with your doctor before undergoing such medications. Spironolactone also causes a significant increase in the production of potassium, though rare, it is a potentially severe side effect that can cause your heart to stop.
You will need to have your potassium levels checked periodically while on this medication.
Natural Effective Testosterone Blockers like Testo Rid contain powerful organic bio-nutrients that work with your body to help block and rid the body of undesirable testosterone levels smoothly and naturally.
Natural testosterone blockers are made from organic materials and trigger less dangerous side effects.
They contain micronutrients and phytonutrients known to inhibit the production of testosterone and promote enzyme activity that converts testosterone to estrogen.
Natural Testosterone Blockers such as Testo Rid is designed to work alone or seamlessly with an estrogen booster to give a smooth, gradual, and comfortable transition.
Natural ingredients like Black Cohosh, Dong Quai, and Saw Palmetto help block, metabolize and rid your body of testosterone at higher consistent levels, naturally and safely.
Transitioning should be as simple, safe, effective, and comfortable as possible. The right testosterone blockers will contribute immensely to achieving that objective.
This is to reduce some of the masculinizing effects of testosterone, reduce some characteristically male traits and aid transgender women in affirming their identity.
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You might also be interested in reading – Male to Female Hormone Replacement Therapy on Natural Hormones
Find out how you can increase estrogen levels fast as a male in our in-depth article “Increase estrogen in males”